Reactions & interactions (36)
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Biochemical Reaction
momelotinib metabolite m5 → momelotinib metabolite m16
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Biochemical Reaction
momelotinib metabolite m19 → momelotinib metabolite m14
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Biochemical Reaction
momelotinib → momelotinib metabolite m5
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Biochemical Reaction
momelotinib metabolite m21 → momelotinib metabolite m8
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Biochemical Reaction
momelotinib metabolite m28 → momelotinib metabolite m14
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Biochemical Reaction
momelotinib → momelotinib metabolite m21
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Biochemical Reaction
momelotinib → momelotinib metabolite m19
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Biochemical Reaction
momelotinib → momelotinib metabolite m16
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Biochemical Reaction
momelotinib metabolite m16 → momelotinib metabolite m17
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Biochemical Reaction
momelotinib metabolite m21 → momelotinib metabolite m28
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Biochemical Reaction
momelotinib metabolite m15 → momelotinib metabolite m8
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Biochemical Reaction
momelotinib → momelotinib metabolite m15
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Catalysis
ABCB1 → Transport
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Catalysis
ABCG2 → Transport
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Catalysis
SLCO1B3 → Transport
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Catalysis
SLCO1B1 → Transport
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Catalysis
CYP2C19 → Biochemical Reaction
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Catalysis
CYP2C8 → Biochemical Reaction
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Catalysis
CYP2C9 → Biochemical Reaction
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Catalysis
CYP3A4 → Biochemical Reaction
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Catalysis
CYP1A2 → Biochemical Reaction
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Catalysis
AOX1 → Biochemical Reaction
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Catalysis
ABCG2 → Transport
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Catalysis
ABCB1 → Transport
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Catalysis
SLCO1B1 → Transport
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Catalysis
SLCO1B3 → Transport
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Inhibition
momelotinib metabolite m21 → JAK1
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Inhibition
momelotinib → JAK2
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Inhibition
momelotinib metabolite m21 → JAK2
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Inhibition
momelotinib → ACVR1
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Inhibition
momelotinib → ABCG2
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Inhibition
momelotinib → JAK1
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Transport
momelotinib → momelotinib
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Transport
momelotinib → momelotinib
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Transport
momelotinib metabolite m21 → momelotinib metabolite m21
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Transport
momelotinib metabolite m21 → momelotinib metabolite m21
Edit history (1)
- 2024-04-22 Create