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PharmGKB · ClinPGx

In Progress: Apatinib Pathway, Pharmacokinetics

PA166319341 Last updated October 2023 Caroline F. Thorn
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Reactions
In Progress: Apatinib Pathway, Pharmacokinetics pathway diagram
In Progress: Apatinib Pathway, Pharmacokinetics — pathway diagram from PharmGKB / ClinPGx
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About this pathway

Work in progress...

Reactions & interactions (24)

  • Biochemical Reaction
    apatinib → apatinib metabolite m1-2
  • Biochemical Reaction
    apatinib metabolite m1-2 → hydroxyapatinib O-glucuronide
  • Biochemical Reaction
    apatinib → apatinib metabolite m1-1
  • Biochemical Reaction
    apatinib metabolite m1-1 → hydroxyapatinib O-glucuronide
  • Biochemical Reaction
    apatinib → apatinib-25-n-oxide
  • Catalysis
    CYP3A4 → Biochemical Reaction
  • Catalysis
    CYP3A5 → Biochemical Reaction
  • Catalysis
    UGT2B7 → Biochemical Reaction
  • Catalysis
    UGT1A1 → Biochemical Reaction
  • Catalysis
    UGT1A4 → Biochemical Reaction
  • Catalysis
    UGT1A9 → Biochemical Reaction
  • Catalysis
    UGT1A8 → Biochemical Reaction
  • Catalysis
    UGT1A3 → Biochemical Reaction
  • Catalysis
    UGT2B4 → Biochemical Reaction
  • Catalysis
    CYP2D6 → Biochemical Reaction
  • Catalysis
    CYP2C9 → Biochemical Reaction
  • Catalysis
    CYP3A4 → Biochemical Reaction
  • Catalysis
    UGT1A4 → Biochemical Reaction
  • Catalysis
    UGT1A1 → Biochemical Reaction
  • Catalysis
    UGT2B7 → Biochemical Reaction
  • Catalysis
    UGT1A3 → Biochemical Reaction
  • Catalysis
    CYP3A5 → Biochemical Reaction
  • Catalysis
    CYP3A4 → Biochemical Reaction
  • Catalysis
    CYP2D6 → Biochemical Reaction

Edit history (1)

  • 2023-10-30 Create
In Progress: Apatinib Pathway, Pharmacokinetics pathway diagram (enlarged)