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PharmGKB · ClinPGx

In Progress: Cabozantinib Pathway, Pharmacokinetics/Pharmacodynamics

PA166306961 Last updated July 2023 Caroline F. Thorn
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Drugs & chemicals
1
Genes
0/0
Conditions
27
Reactions
In Progress: Cabozantinib Pathway, Pharmacokinetics/Pharmacodynamics pathway diagram
In Progress: Cabozantinib Pathway, Pharmacokinetics/Pharmacodynamics — pathway diagram from PharmGKB / ClinPGx
Click to enlarge

About this pathway

Work in progress...

Reactions & interactions (27)

  • Biochemical Reaction
    cabozantinib cabozantinib n-oxide
  • Biochemical Reaction
    cabozantinib cabozantinib metabolite m7
  • Biochemical Reaction
    cabozantinib metabolite m7 cabozantinib metabolite m2a
  • Biochemical Reaction
    cabozantinib cabozantinib metabolite m9
  • Catalysis
    ABCC2 Transport
  • Catalysis
    ABCG2 Transport
  • Catalysis
    SLCO1B1 Transport
  • Catalysis
    SLCO1B3 Transport
  • Catalysis
    ABCC2 Transport
  • Catalysis
    CYP2C9 Biochemical Reaction
  • Catalysis
    CYP3A4 Biochemical Reaction
  • Inhibition
    cabozantinib n-oxide CYP2C8
  • Inhibition
    cabozantinib MET
  • Inhibition
    cabozantinib CYP2C8
  • Inhibition
    cabozantinib AXL
  • Inhibition
    cabozantinib metabolite m2a SLC22A6
  • Inhibition
    cabozantinib KDR
  • Inhibition
    cabozantinib ABCB1
  • Inhibition
    cabozantinib SLC47A2
  • Inhibition
    cabozantinib metabolite m2a SLC47A2
  • Inhibition
    cabozantinib RET
  • Inhibition
    cabozantinib metabolite m2a ABCB11
  • Inhibition
    cabozantinib SLC47A1
  • Inhibition
    cabozantinib metabolite m2a SLC22A8
  • Inhibition
    cabozantinib metabolite m2a SLC47A1
  • Transport
    cabozantinib cabozantinib
  • Transport
    cabozantinib metabolite m2a cabozantinib metabolite m2a

Edit history (1)

  • 2023-07-17 Create
In Progress: Cabozantinib Pathway, Pharmacokinetics/Pharmacodynamics pathway diagram (enlarged)